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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T6380 | AMG 900 | AMG900,AMG-900 | p38 MAPK , Tyrosine Kinases , Aurora Kinase |
AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/C with IC50 of 5 nM/4 nM /1 nM. It is >10-fold selective for Aurora kinases than p38α, Tyk2, JNK2, Met and Tie2. Phase 1. |